143824-77-5

  • Product Name:FMOC-ARG(BOC)2-OH
  • Molecular Formula:C31H40 N4 O8
  • Molecular Weight:596.681
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Product Details

Purity:99%

Cost-effective and customizable FMOC-ARG(BOC)2-OH 143824-77-5 in stock

  • Molecular Formula:C31H40 N4 O8
  • Molecular Weight:596.681
  • PKA:3.80±0.21(Predicted) 
  • PSA:167.35000 
  • Density:1.255g/cm3 
  • LogP:6.33660 

FMOC-ARG(BOC)2-OH(Cas 143824-77-5) Usage

InChI:InChI=1/C31H40N4O8/c1-30(2,3)42-28(39)34-26(35-29(40)43-31(4,5)6)32-17-11-16-24(25(36)37)33-27(38)41-18-23-21-14-9-7-12-19(21)20-13-8-10-15-22(20)23/h7-10,12-15,23-24H,11,16-18H2,1-6H3,(H,33,38)(H,36,37)(H2,32,34,35,39,40)/t24-/m0/s1

143824-77-5 Relevant articles

Modular Solid-Phase Synthesis of Antiprotozoal Barnesin Derivatives

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Here, we applied and optimized a solid s...

An efficient and economical method for the preparation of Fmoc-Arg ωω (Boc) 2-OH

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143824-77-5 Process route

Nα-benzyloxycarbonyl-L-ornithine
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Nα-benzyloxycarbonyl-L-ornithine

Fmoc-Arg<sup>ω,ω'</sup>(Boc)2-OH
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Fmoc-Argω,ω'(Boc)2-OH

Conditions
Conditions Yield
Multi-step reaction with 3 steps
1: Triton-B / methanol; dimethylsulfoxide / 40 h / 10 °C
2: 99 percent / hydrogen / 10percent Pd/C / methanol / 0.67 h / 1551.4 Torr
3: 99.6 percent / DIPEA / CH2Cl2 / 1.17 h
With hydrogen; N-benzyl-trimethylammonium hydroxide; N-ethyl-N,N-diisopropylamine; palladium on activated charcoal; In methanol; dichloromethane; dimethyl sulfoxide;
9-fluorenylmethyl N-succinimidyl carbonate
102774-86-7

9-fluorenylmethyl N-succinimidyl carbonate

H-L-Arg(Boc)<SUB>2</SUB>-OH
145315-38-4

H-L-Arg(Boc)2-OH

N-α-(9-fluorenylmethyloxycarbonyl)-N-ω′,N-ω″-bis-tert-butyloxycarbonyl-L-argine
143824-77-5

N-α-(9-fluorenylmethyloxycarbonyl)-N-ω′,N-ω″-bis-tert-butyloxycarbonyl-L-argine

Conditions
Conditions Yield
With ethylenediaminetetraacetic acid; sodium hydrogencarbonate; In acetone; at 20 ℃;
84%

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